Mitochondrial Β· LongevityTier 3 β€” Animal + early human data

MOTS-c

Mitochondrial Open Reading Frame of the 12S rRNA-c

Mitochondria-derived peptide that acts as a metabolic regulator, improving insulin sensitivity and exercise capacity. Circulating levels naturally decline with age.

πŸ’‰ SC injection🧊 Lyophilised: refrigerate; reconstituted: refrigerate, use within 30 days

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Mechanism of Action

Translocates to the nucleus and mitochondria, activating AMPK and FOXO pathways, upregulating GLUT4, reducing ROS production, and enhancing mitochondrial biogenesis.

Clinical Applications

  • βœ“Metabolic health and insulin sensitivity
  • βœ“Anti-aging and longevity
  • βœ“Exercise performance enhancement
  • βœ“Age-related muscle loss (sarcopenia)
  • βœ“Obesity-related metabolic dysfunction

Dosing Protocol

Recommended Dosing

SC injection. 5–10 mg, 2–3x per week. Often dosed before exercise. Cycles of 8–12 weeks. Research compound β€” human data limited.

Safety & Contraindications

Possible Side Effects

  • ⚠Largely unknown β€” limited human data
  • ⚠Injection site reactions
  • ⚠Possible excessive hypoglycaemia if combined with insulin

Contraindications

  • βœ•Pregnancy
  • βœ•Known diabetes on insulin (hypoglycaemia risk)

Combinations & Synergies

πŸ”— Humaninsynergistic mitochondrial protection
πŸ”— 5-Amino-1MQcomplementary metabolic activation
πŸ”— Epithalonlongevity stack