GH Secretagogues Β· RegenerativeTier 2 β€” Good human studies

Hexarelin

Examorelin Β· EP 23905

The most potent GHRP class peptide for GH release, with additional cardioprotective effects via CD36 receptors. Significant desensitization occurs with continuous use.

πŸ’‰ SC injection🧊 Lyophilised: refrigerate; reconstituted: refrigerate, use within 30 days

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Mechanism of Action

Potent GHSR-1a agonist producing maximal GH pulses. Also binds cardiac CD36 receptors independent of GH, providing direct cardioprotective and anti-fibrotic effects.

Clinical Applications

  • βœ“Maximum GH stimulation
  • βœ“Cardiac protection and post-MI recovery
  • βœ“Short-burst protocols for peak GH testing
  • βœ“Body composition in experienced users

Dosing Protocol

Recommended Dosing

SC injection. 100–200 mcg, 1–3x daily. Use in short cycles (4–6 weeks) to avoid desensitization. Allow at least equal off-time.

Safety & Contraindications

Possible Side Effects

  • ⚠Rapid desensitization with continuous use
  • ⚠Strong cortisol and prolactin elevation
  • ⚠Water retention
  • ⚠Significant hunger
  • ⚠Lethargy

Contraindications

  • βœ•Active malignancy
  • βœ•Elevated prolactin baseline
  • βœ•Pregnancy
  • βœ•Diabetes

Combinations & Synergies

πŸ”— CJC-1295maximum GH amplification (advanced protocols only)