NeuralTier 3 β€” Animal + early human data

DSIP

Delta Sleep-Inducing Peptide Β· DSIP nonapeptide

Endogenous nonapeptide that modulates sleep architecture, particularly promoting slow-wave (delta) sleep. Also shows stress-regulatory and mild analgesic properties. Blood-brain barrier permeable.

πŸ’‰ SC injection🧊 Lyophilised: room temperature. Reconstituted: refrigerate (2–8 Β°C), use within 14 days. Protect from light and heat.

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Mechanism of Action

DSIP modulates GABAergic and glutamatergic neurotransmission in the thalamo-cortical sleep circuits. Inhibits CRH secretion and reduces ACTH/cortisol at night, facilitating sleep onset. Crosses the BBB intact due to its small size and lipophilic character.

Clinical Applications

  • βœ“Insomnia and sleep-onset difficulties
  • βœ“Improving slow-wave (deep) sleep fraction
  • βœ“Stress-related sleep disruption and HPA axis dysregulation
  • βœ“Withdrawal support (opiate, alcohol) β€” limited evidence
  • βœ“Circadian rhythm re-synchronisation (shift work, jet lag)

Dosing Protocol

Recommended Dosing

SC injection. 100–200 mcg, 20–30 min before desired sleep onset. Typical cycle: 5 nights on, 2 nights off, for 4–8 weeks. Some protocols use 100 mcg + Epithalon 10 mg as a sleep stack.

Safety & Contraindications

Possible Side Effects

  • ⚠Morning grogginess if dose is too high or timed poorly
  • ⚠Mild dizziness shortly after injection
  • ⚠Vivid dreams (generally non-distressing)

Contraindications

  • βœ•Sleep apnoea (undiagnosed/untreated) β€” deepening sleep may worsen apnoea events
  • βœ•Pregnancy
  • βœ•Operating machinery or driving same evening

Combinations & Synergies

πŸ”— Epithaloncomplementary sleep/longevity stack β€” DSIP for sleep onset, Epithalon for circadian clock normalisation
πŸ”— MK-677oral GH secretagogue before bed synergises with DSIP-promoted deep sleep for GH pulse optimisation
πŸ”— Selankif anxiety is the primary driver of insomnia, Selank intranasal + DSIP SC addresses both axes